SCHEMBL7069604

SCHEMBL7069604

Cc1cccc(NC(=O)C(C)(O)CS(=O)(=O)c2ccc(F)cc2)c1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 4/20 0.62
CYP3A4 P08684 3/20 0.62
CYP2C9 P11712 2/20 0.62
ALDH1A1 P00352 2/20 0.62
HPGD P15428 2/20 0.62
AR P10275 11/20 0.61
ABCB11 O95342 1/20 0.60
ALB P02768 1/20 0.60
PGR P06401 1/20 0.60
ADRA2C P18825 1/20 0.60
GHSR Q92847 1/20 0.60
CYP2D6 P10635 1/20 0.54
KDM4E B2RXH2 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18720887 1.00 CYP2C19 (0.62) CYP2C19CYP3A4CYP2C9ALDH1A1HPGD
SCHEMBL17381289 0.86 CYP2C19 (0.83) CYP2C19CYP3A4CYP2C9ALDH1A1HPGD
SCHEMBL4620937 0.86 CYP2C19 (0.83) CYP2C19CYP3A4CYP2C9ALDH1A1HPGD
SCHEMBL7074011 0.85 AR (0.62) CYP2C19CYP3A4CYP2C9ALDH1A1HPGD
SCHEMBL18720886 0.84 AR (0.77) CYP2C19CYP3A4CYP2C9ALDH1A1HPGD
SCHEMBL6769180 0.82 GHSR (0.53) CYP2C19CYP3A4CYP2C9ALDH1A1HPGD
SCHEMBL18720880 0.81 AR (0.66) CYP2C19CYP3A4CYP2C9ALDH1A1HPGD
SCHEMBL17381241 0.81 AR (0.74) CYP2C19ARABCB11ALBPGR
SCHEMBL14559210 0.81 AR (0.74) CYP2C19ARABCB11ALBPGR
SCHEMBL18720853 0.80 AR (0.67) CYP2C19CYP3A4CYP2C9ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003043630-A1 SOLID PHARMACEUTICAL COMPOSITION COMPRISING 4-CYANO-TRIFLUORO-3-(4-FLUOROPHENYL SULPHONYL)-2-HYDROXY-2-METHYLPROPIONO- M TOLUIDIDE, PVP, AN ANTI-OESTROGEN AND/OR AN AROMATASE INHIBITOR ASTRAZENECA UK LIMITED (GB) 2003-05-30 WO claimed