SCHEMBL7069709

SCHEMBL7069709

Cc1nc(COc2cncc(C(=Cc3ccncc3)c3ccncc3)c2)c[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.36
CYP11B2 P19099 1/20 0.36
SIRT2 Q8IXJ6 2/20 0.35
SIRT1 Q96EB6 2/20 0.35
SIRT3 Q9NTG7 2/20 0.35
MAPK1 P28482 3/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
AKT1 P31749 13/20 0.33
CLK4 Q9HAZ1 6/20 0.33
PRKACA P17612 6/20 0.33
ROCK2 O75116 5/20 0.33
MAP4K4 O95819 5/20 0.33
ROCK1 Q13464 5/20 0.33
DYRK1A Q13627 5/20 0.33
PKN2 Q16513 5/20 0.33
MKNK2 Q9HBH9 5/20 0.33
STK17A Q9UEE5 5/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6833433 0.72 AKT1 (0.60) CYP19A1CYP11B2SIRT2SIRT1SIRT3
Hydrochloric Acid SCHEMBL6931715 0.66 AKT1 (0.67) CYP19A1CYP11B2MAPK1AKT1CLK4
SCHEMBL13141937 0.61 CYP19A1 (0.72) CYP19A1CYP11B2KDM4EMAPTKMT2A
SCHEMBL6931724 0.60 CYP11B2 (0.44) CYP19A1CYP11B2AKT1CLK4PRKACA
SCHEMBL16946606 0.57 CYP19A1 (1.00) CYP19A1CYP11B2LMNAMAPTKMT2A
SCHEMBL19046336 0.57
SCHEMBL7691608 0.57 AKT1 (0.59) KDM4EAKT1CLK4PRKACAROCK2
SCHEMBL7691611 0.57 AKT1 (0.59) KDM4EAKT1CLK4PRKACAROCK2
SCHEMBL23332034 0.56 CYP19A1 (0.73) CYP19A1CYP11B2MAPK1MAPTKMT2A
SCHEMBL23332031 0.56 CYP19A1 (0.79) CYP19A1CYP11B2MAPK1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1463505-A2 3-(PHENYL-ALKOXY)-5-(PHENYL)-PYRIDINE DERIVATIVES AND RELATED COMPOUNDS AS KINASE INHIBITORS FOR THE TREATMENT OF CANCER Abbott Laboratories (US) 2004-10-06 EP disclosed
WO-2003051366-A2 3-(PHENYL-ALKOXY)-5-(PHENYL)-PYRIDINE DERIVATIVES AND RELATED COMPOUNDS AS KINASE INHIBITORS FOR THE TREATMENT OF CANCER ABBOTT LABORATORIES (US) 2003-06-26 WO disclosed