SCHEMBL707064

SCHEMBL707064

O=C(NN1C(=O)[C@@H]2[C@H]3C=C[C@H]([C@@H]4C[C@H]34)[C@@H]2C1=O)c1ccccc1C(F)(F)F

nearest known ligand 0.69

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
ALDH1A1 P00352 4/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
GAA P10253 2/20 0.47
LMNA P02545 2/20 0.46
MAPT P10636 1/20 0.42
CYP3A4 P08684 1/20 0.41
HTT P42858 1/20 0.40
MAPK1 P28482 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10029229 0.81 MEN1 (0.74) MEN1KMT2AALDH1A1SMN1; SMN2GAA
SCHEMBL10029222 0.81 KMT2A (0.60) MEN1KMT2AALDH1A1SMN1; SMN2GAA
Tecovirimat SCHEMBL20126651 0.79 ALDH1A1 (0.73) MEN1KMT2AALDH1A1SMN1; SMN2GAA
Tecovirimat SCHEMBL10034023 0.79 ALDH1A1 (0.73) MEN1KMT2AALDH1A1SMN1; SMN2GAA
Tecovirimat SCHEMBL16177983 0.79 ALDH1A1 (0.73) MEN1KMT2AALDH1A1SMN1; SMN2GAA
Tecovirimat SCHEMBL14601849 0.79 ALDH1A1 (0.73) MEN1KMT2AALDH1A1SMN1; SMN2GAA
Tecovirimat SCHEMBL404303 0.79 ALDH1A1 (0.73) MEN1KMT2AALDH1A1SMN1; SMN2GAA
SCHEMBL18691802 0.78 ALDH1A1 (0.76) MEN1KMT2AALDH1A1SMN1; SMN2GAA
SCHEMBL405810 0.74 ALDH1A1 (0.76) MEN1KMT2AALDH1A1SMN1; SMN2GAA
SCHEMBL25239750 0.72 PTGS1 (0.63) MEN1KMT2AALDH1A1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638938-B1 COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATMENT AND PREVENTION OF ORTHOPOXVIRUS INFECTIONS AND ASSOCIATED DISEASES SIGA TECH INC (US) 2017-04-12 EP claimed
US-8124643-B2 Compounds, compositions and methods for treatment and prevention of orthopoxvirus infections and associated diseases SIGA TECHNOLOGIES, INC. (US) 2012-02-28 US claimed
US-8039504-B2 heating a mixture of anti-tricyclo[3.2.2.0]non-6-ene-endo-8, endo-9-dicarboxylic acid anhydride, 4-(trifluoromethyl)benzhydrazide, and ethanol at reflux, concetrating and recrystallizing; 4-Trifluoromethyl-N- (3,3a,4,4a,5,5a,6,6a,- octahydro-1,3-dioxo-4,6- ethenocycloprop[f]isoindol- 2(1H)-yl)-benzamide SIGA TECHNOLOGIES, INC. (US) 2011-10-18 US claimed