SCHEMBL7073105

SCHEMBL7073105

CNc1ccccc1C(=O)NCCN1CC2CC(c3ccc(F)cc3)C2C1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.45
PLD1 Q13393 5/20 0.44
CRBN Q96SW2 1/20 0.44
BCL3 P20749 4/20 0.43
ALDH1A1 P00352 3/20 0.42
PKM P14618 1/20 0.42
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PLD2 O14939 2/20 0.39
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7078371 0.90 CRBN (0.44) PLD1CRBNBCL3ALDH1A1PLD2
SCHEMBL7774070 0.87 PLD1 (0.44) KDM4EPLD1BCL3ALDH1A1GAA
SCHEMBL7074973 0.86 KDM4E (0.44) KDM4EPLD1BCL3ALDH1A1HPGD
SCHEMBL8882719 0.84 HPGD (0.52) PLD1HPGD
SCHEMBL7774077 0.83 PLD1 (0.53) PLD1ALDH1A1PLD2
SCHEMBL7781108 0.82 PLD1 (0.53) PLD1PLD2
SCHEMBL8876709 0.82 EPHX2 (0.41) PLD1BCL3PLD2
SCHEMBL8989699 0.81 PLD1 (0.56) PLD1ALDH1A1PLD2
Cyclopropane SCHEMBL7076457 0.79 PLD1 (0.41) PLD1PLD2KMT2A
Cyclopentane SCHEMBL7071125 0.79 PLD1 (0.41) PLD1PLD2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0740658-B1 N-SUBSTITUTED AZABICYCLOHEPTANE DERIVATIVES USED, FOR EXAMPLE, AS NEUROLEPTICS ABBOTT GMBH & CO KG (DE) 2003-07-02 EP disclosed
US-5616705-A N-substituted azabicycloheptane derivatives, their preparation and use BASF AKTIENGESELLSCHAFT (DE) 1997-04-01 US disclosed