SCHEMBL7074973

SCHEMBL7074973

Nc1ccccc1C(=O)NCCN1CC2CC(c3ccc(F)cc3)C2C1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 1/20 0.44
PLD1 Q13393 2/20 0.44
ADRA1B P35368 1/20 0.42
KDM1A O60341 3/20 0.39
HPGD P15428 1/20 0.39
BCL3 P20749 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7075387 0.90 ALDH1A1 (0.44) KDM4EALDH1A1LMNAADRA1BHPGD
SCHEMBL7774070 0.89 PLD1 (0.44) KDM4EALDH1A1PLD1HPGDBCL3
SCHEMBL8882719 0.86 HPGD (0.52) PLD1KDM1AHPGD
SCHEMBL7073105 0.86 KDM4E (0.45) KDM4EALDH1A1PLD1HPGDBCL3
SCHEMBL7774077 0.85 PLD1 (0.53) ALDH1A1PLD1KDM1A
SCHEMBL7781108 0.84 PLD1 (0.53) PLD1KDM1A
SCHEMBL8876709 0.83 EPHX2 (0.41) LMNAPLD1ADRA1BKDM1ABCL3
SCHEMBL8989699 0.83 PLD1 (0.56) ALDH1A1PLD1KDM1A
Cyclopropane SCHEMBL7076457 0.81 PLD1 (0.41) PLD1
Cyclopentane SCHEMBL7071125 0.81 PLD1 (0.41) PLD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0740658-B1 N-SUBSTITUTED AZABICYCLOHEPTANE DERIVATIVES USED, FOR EXAMPLE, AS NEUROLEPTICS ABBOTT GMBH & CO KG (DE) 2003-07-02 EP disclosed
US-5616705-A N-substituted azabicycloheptane derivatives, their preparation and use BASF AKTIENGESELLSCHAFT (DE) 1997-04-01 US disclosed
EP-0740658-A1 N-SUBSTITUTED AZABICYCLOHEPTANE DERIVATIVES USED, FOR EXAMPLE, AS NEUROLEPTICS BASF AKTIENGESELLSCHAFT (DE) 1996-11-06 EP disclosed
WO-1995015312-A1 N-SUBSTITUTED AZABICYCLOHEPTANE DERIVATIVES USED, FOR EXAMPLE, AS NEUROLEPTICS BASF AKTIENGESELLSCHAFT (DE) 1995-06-08 WO disclosed