SCHEMBL7076065

SCHEMBL7076065

CC(C(=O)O)c1cc(N)cc(C(C)C(=O)O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.45
PTGS1 P23219 10/20 0.43
CXCR1 P25024 4/20 0.43
CXCR2 P25025 4/20 0.43
LMNA P02545 3/20 0.43
SLC22A6 Q4U2R8 3/20 0.43
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
PMP22 Q01453 2/20 0.43
CXCL8 P10145 2/20 0.43
RECQL P46063 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 1/20 0.43
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
THPO P40225 1/20 0.43
HIF1A Q16665 1/20 0.43
AKR1C3 P42330 8/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL999861 0.95 PTGS2 (0.45) PTGS2PTGS1CXCR1CXCR2LMNA
SCHEMBL7080519 0.80 NPC1 (0.46) LMNAMAPTSMN1; SMN2ALDH1A1CYP3A4
SCHEMBL1001487 0.80 PTGS2 (0.44) PTGS2PTGS1CXCR1CXCR2LMNA
SCHEMBL8579553 0.79 PTGS1 (0.59) PTGS2PTGS1CXCR1CXCR2LMNA
SCHEMBL360725 0.79 PTGS1 (0.59) PTGS2PTGS1CXCR1CXCR2LMNA
SCHEMBL8960142 0.79 PTGS2 (0.54) PTGS2PTGS1CXCR1CXCR2LMNA
SCHEMBL5846200 0.79 PTGS2 (0.54) PTGS2PTGS1CXCR1CXCR2LMNA
Hydrochloric Acid SCHEMBL1177638 0.78 PTGS1 (0.57) PTGS2PTGS1CXCR1CXCR2LMNA
SCHEMBL2818028 0.77 PTGS2 (0.61) PTGS2PTGS1CXCR1CXCR2LMNA
SCHEMBL2852282 0.77 PTGS2 (0.61) PTGS2PTGS1CXCR1CXCR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1013636-B1 Preparation of allylic aromatic compounds AMERSHAM HEALTH AS (NO) 2003-07-09 EP disclosed
US-6284894-B1 AROMATIC AMINE IS REACTED FIRST WITH A NITRITE AND THEN WITH AN ALLYLIC OLEFIN HAVING AN ELIMINATABLE TERMINAL SUBSTITUENT. NYCOMED IMAGING AS (NO) 2001-09-04 US disclosed
EP-1013636-A1 Preparation of allylic aromatic compounds NYCOMED IMAGING AS (NO) 2000-06-28 EP disclosed