SCHEMBL7076733

SCHEMBL7076733

Clc1ccc(-n2cnc3c(-c4ccco4)nc([AsH2])nc32)cc1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.59
ADORA1 P30542 7/20 0.43
XDH P47989 1/20 0.42
PI4KA P42356 1/20 0.40
PI4K2B Q8TCG2 1/20 0.40
PI4K2A Q9BTU6 1/20 0.40
PI4KB Q9UBF8 1/20 0.40
PIK3R1 P27986 1/20 0.39
PIK3CA P42336 1/20 0.39
PTGS1 P23219 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939895 0.74 ADORA2A (0.75) ADORA2AADORA1XDH
SCHEMBL5462775 0.69 ADORA2A (0.79) ADORA2AADORA1
SCHEMBL6944247 0.69 ADORA2A (0.53) ADORA2AADORA1PIK3R1PIK3CA
SCHEMBL3269621 0.68 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL3269358 0.65 ADORA2A (0.82) ADORA2AADORA1
SCHEMBL5451859 0.65 ADORA2A (0.70) ADORA2AADORA1PI4KAPI4K2BPI4K2A
SCHEMBL3267606 0.64 ADORA2A (0.56) ADORA2AADORA1
SCHEMBL3273422 0.63 ADORA2A (0.83) ADORA2AADORA1
SCHEMBL1653877 0.63 ADORA2A (0.77) ADORA2AADORA1
SCHEMBL3268990 0.62 CCNE1 (0.45) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed