SCHEMBL6944247

SCHEMBL6944247

O=S(=O)=Nc1nc(-c2ccco2)c2ncn(-c3ccc(Br)cc3)c2n1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.53
ADORA1 P30542 12/20 0.36
APOBEC3G Q9HC16 1/20 0.35
PIK3R1 P27986 1/20 0.35
PIK3CA P42336 1/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA2B P29275 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6949760 0.73 ADORA2A (0.41) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL7076733 0.69 ADORA2A (0.59) ADORA2AADORA1PIK3R1PIK3CA
SCHEMBL6939895 0.65 ADORA2A (0.75) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3267809 0.63 ADORA2A (0.56) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL23436456 0.59 XDH (0.49) ADORA2A
SCHEMBL3269891 0.58 ADORA2A (0.58) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3270277 0.58 ADORA2A (0.76) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3267606 0.58 ADORA2A (0.56) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3269113 0.58 ADORA2A (0.77) ADORA2AADORA1
SCHEMBL3310025 0.58 XDH (0.76)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP claimed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO claimed