SCHEMBL7078618

SCHEMBL7078618

CC(=O)Oc1nc(C(C)C)c(Sc2cccc([N+](=O)[O-])c2)n1Cc1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.42
S1PR3 Q99500 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
GNRHR P30968 1/20 0.36
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 6/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPK1 P28482 1/20 0.35
CTSD P07339 1/20 0.35
ACHE P22303 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084592 0.88 CFTR (0.41) CFTRS1PR3CYP1A2CYP3A4GNRHR
SCHEMBL8800655 0.87 CFTR (0.41) CFTRS1PR3CYP1A2CYP3A4GNRHR
SCHEMBL7084768 0.87 PTGDR2 (0.36) CYP1A2MAPTPKML3MBTL1KDM4E
SCHEMBL6973925 0.86 PDE4A (0.37) GNRHRMAPTLMNAPKML3MBTL1
SCHEMBL7081438 0.86 TP53 (0.36) MAPTPKML3MBTL1KDM4EKMT2A
SCHEMBL6973156 0.86 S1PR3 (0.38) S1PR3MAPTKDM4EKMT2A
SCHEMBL7084512 0.86 IRAK4 (0.38) CFTRCYP1A2CYP3A4MAPTLMNA
SCHEMBL6972280 0.85 CFTR (0.40) CFTRS1PR3CYP1A2CYP3A4GNRHR
SCHEMBL6972931 0.84 CFTR (0.44) CFTRS1PR3CYP1A2CYP3A4GNRHR
SCHEMBL6961923 0.84 CYP1A2 (0.44) CFTRS1PR3CYP1A2CYP3A4GNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed