SCHEMBL7079167

SCHEMBL7079167

CCCCCCn1c(CCO)nc(C(C)C)c1Sc1cc(C)cc(C)c1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GCGR P47871 12/20 0.34
TSSK1B Q9BXA7 1/20 0.33
TLR7 Q9NYK1 1/20 0.32
TLR8 Q9NR97 2/20 0.31
TP53 P04637 2/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976885 0.96 MEN1 (0.33) GCGRMAPT
SCHEMBL6962650 0.95 TLR7 (0.35) GCGRTSSK1BTLR7TLR8TP53
SCHEMBL6966535 0.91 GCGR (0.35) GCGRTSSK1BTLR8
SCHEMBL6966167 0.91 ALDH1A1 (0.36) MAPT
SCHEMBL7081111 0.90 MEN1 (0.32) GCGRTLR7HDAC1HDAC8MAPT
SCHEMBL7080973 0.88 HSP90B1 (0.38) GCGRTLR7MAPT
SCHEMBL6965442 0.88 GCGR (0.36) GCGRTLR7TP53
SCHEMBL6972574 0.87 ALDH1A1 (0.35) GCGRMAPT
SCHEMBL6973709 0.86 GCGR (0.34) GCGRMAPT
SCHEMBL6960610 0.86

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed