SCHEMBL7080717

SCHEMBL7080717

Nc1nc(NC2CCCCC2)nc(N2CCCCC2)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.65
SMN1; SMN2 Q16637 2/20 0.65
NPSR1 Q6W5P4 2/20 0.65
CTSL P07711 1/20 0.52
CTSB P07858 1/20 0.52
CTSS P25774 1/20 0.52
CTSK P43235 1/20 0.52
MEN1 O00255 1/20 0.52
ALDH1A1 P00352 1/20 0.52
MAPT P10636 1/20 0.52
MAPK1 P28482 1/20 0.52
BLM P54132 1/20 0.52
KMT2A Q03164 1/20 0.52
NUDT1 P36639 1/20 0.49
ATM Q13315 1/20 0.48
LMNA P02545 1/20 0.46
HPGD P15428 1/20 0.46
ROCK1 Q13464 1/20 0.46
HRH4 Q9H3N8 2/20 0.45
CNR2 P34972 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14504424 0.90 SMN1; SMN2 (0.72) HTTSMN1; SMN2NPSR1CTSLCTSB
SCHEMBL14504419 0.90 SMN1; SMN2 (0.72) HTTSMN1; SMN2NPSR1CTSLCTSB
SCHEMBL14504177 0.90 SMN1; SMN2 (0.72) HTTSMN1; SMN2NPSR1CTSLCTSB
SCHEMBL8051814 0.90 HTT (0.72) HTTSMN1; SMN2NPSR1CTSLCTSB
SCHEMBL2241510 0.83 HTT (0.48) HTTSMN1; SMN2NPSR1CTSLCTSB
SCHEMBL2241516 0.83 HTT (0.48) HTTSMN1; SMN2NPSR1CTSLCTSB
SCHEMBL12757927 0.83 HTT (0.68) HTTSMN1; SMN2NPSR1CTSLCTSB
SCHEMBL6272713 0.83 SMN1; SMN2 (0.63) HTTSMN1; SMN2NPSR1CTSLCTSB
SCHEMBL6640516 0.82 PDE4A (0.55) HTTSMN1; SMN2NPSR1NUDT1HRH4
SCHEMBL2783836 0.82 NUDT1 (0.51) HTTSMN1; SMN2NPSR1CTSKMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030148269-A1 Centrifugally-enhanced method of determining ligand/target affinity HOLZMAN THOMAS F (US) 2003-08-07 US disclosed
EP-1161684-A1 CENTRIFUGALLY-ENHANCED METHOD OF DETERMINING LIGAND/TARGET AFFINITY ABBOTT LABORATORIES (US) 2001-12-12 EP disclosed
WO-2000055625-A1 CENTRIFUGALLY-ENHANCED METHOD OF DETERMINING LIGAND/TARGET AFFINITY ABBOTT LABORATORIES (US) 2000-09-21 WO disclosed