SCHEMBL7080920

SCHEMBL7080920

CC(C)(C)OC(=O)N1CCC(c2ccc(OCCOc3ccccc3)cc2)C(OCc2ccc3ccccc3c2)C1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
REN P00797 15/20 0.55
PRMT5 O14744 1/20 0.45
YAP1 P46937 2/20 0.45
TACR1 P25103 1/20 0.44
PDE4B Q07343 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6041532 0.92 REN (0.47) RENPRMT5YAP1TACR1
SCHEMBL6042241 0.90 REN (0.49) RENPRMT5YAP1TACR1
SCHEMBL6041545 0.90 REN (0.47) RENPRMT5YAP1TACR1
SCHEMBL6043110 0.89 REN (0.46) RENPRMT5YAP1TACR1
SCHEMBL6042351 0.89 REN (0.46) RENPRMT5YAP1TACR1
SCHEMBL6042535 0.89 REN (0.53) RENYAP1
SCHEMBL7562146 0.89 REN (0.48) RENPRMT5YAP1TACR1
SCHEMBL6042529 0.89 REN (0.59) REN
SCHEMBL6043910 0.88 REN (0.55) RENPRMT5YAP1
SCHEMBL7080924 0.87 REN (0.54) REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863875-B1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY HOFFMANN LA ROCHE (CH) 2003-06-04 EP disclosed
EP-0863875-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1998-09-16 EP disclosed
WO-1997009311-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1997-03-13 WO disclosed