SCHEMBL7083004

SCHEMBL7083004

Cc1cc(C)cc(Sc2[nH]c(C(O)Cc3ccncc3)nc2C(C)C)c1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.32
GAA P10253 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
POLB P06746 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6967546 0.90 IDO1 (0.38) POLBKMT2A
SCHEMBL6960986 0.88 GSK3B (0.32) GSK3BCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6973238 0.88 CYP1A2 (0.33) GSK3BCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6970549 0.87 IDO1 (0.35) CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7078351 0.86 SLC6A4 (0.36) GSK3BGAACYP1A2CYP3A4CYP2C9
SCHEMBL6976919 0.83
SCHEMBL8109549 0.83 MAPK14 (0.34) GSK3BCYP3A4
SCHEMBL7081552 0.83 PTPRA (0.34) CYP1A2CYP3A4CYP2C9CYP2C19KMT2A
SCHEMBL7079911 0.83 SLC2A1 (0.34) POLBMEN1KMT2A
Carbamic Acid SCHEMBL4573817 0.82 CDC7 (0.33) GSK3BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed