SCHEMBL8109549

SCHEMBL8109549

CC(C)c1nc(C(O)Cc2ccncc2)[nH]c1Sc1cccc(F)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.34
MAPK13 O15264 2/20 0.34
MAPK12 P53778 2/20 0.34
MAPK11 Q15759 2/20 0.34
CYP17A1 P05093 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
HAO1 Q9UJM8 1/20 0.32
ROCK1 Q13464 3/20 0.32
TYMS P04818 1/20 0.32
ALOX5 P09917 1/20 0.32
SLC6A9 P48067 4/20 0.32
TP53 P04637 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
RAF1 P04049 1/20 0.31
PDE4A P27815 1/20 0.31
NPC1 O15118 1/20 0.30
GSK3B P49841 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6960986 0.90 GSK3B (0.32) CYP3A4GSK3BROCK2
SCHEMBL7083467 0.89 IDO1 (0.35) CYP3A4HAO1TP53RAB9ASMN1; SMN2
SCHEMBL7079911 0.88 SLC2A1 (0.34) TYMSSLC6A9TP53RAB9ASMN1; SMN2
SCHEMBL7078351 0.87 SLC6A4 (0.36) MAPK14MAPK13MAPK12MAPK11CYP3A4
SCHEMBL7079967 0.86 GCGR (0.36) HAO1TYMSSLC6A9
SCHEMBL6973954 0.86 ROCK1 (0.32) MAPK14MAPK13MAPK12MAPK11ROCK1
SCHEMBL6967986 0.85 SLC6A9 (0.34) MAPK14HAO1TYMSSLC6A9RAB9A
SCHEMBL7084286 0.85 MAPK13 (0.30) MAPK14MAPK13MAPK12MAPK11
SCHEMBL6974320 0.83 MAPK14 (0.34) MAPK14MAPK13MAPK12MAPK11CYP17A1
SCHEMBL6963027 0.83 ALOX5 (0.38) CYP3A4ALOX5RAB9APDE4ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed