SCHEMBL7083271

SCHEMBL7083271

CO/N=C1\C[C@@H](C(=O)NC[C@H](O)c2ccccc2)N(C(=O)c2ccc(-c3ccccc3)c(C)c2)C1

nearest known ligand 0.83

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OXTR P30559 5/20 0.83
AVPR1A P37288 3/20 0.83
ROCK2 O75116 4/20 0.39
ROCK1 Q13464 4/20 0.39
ADRB1 P08588 2/20 0.37
ADRB3 P13945 2/20 0.37
PRSS1 P07477 1/20 0.36
MMP1 P03956 1/20 0.34
MMP3 P08254 1/20 0.34
MMP7 P09237 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
AGTR1 P30556 2/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4945458 1.00 OXTR (0.83) OXTRAVPR1AROCK2ROCK1ADRB1
SCHEMBL7219611 0.91 OXTR (0.79) OXTRAVPR1AROCK2ROCK1ADRB1
SCHEMBL4936354 0.91 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL4936174 0.91 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL4942975 0.91 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL5743780 0.91 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL4943198 0.91 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL5743785 0.91 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL4940385 0.91 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL4936543 0.91 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268418-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS Applied Research Systems ARS Holding N.V. (AN) 2003-01-02 EP claimed
WO-2001074769-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-11 WO claimed