SCHEMBL7083517

SCHEMBL7083517

CC(C)c1nc(CCCO)n(C)c1Sc1cccc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GCGR P47871 3/20 0.38
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
NOTUM Q6P988 1/20 0.33
DHODH Q02127 1/20 0.32
HAO1 Q9UJM8 1/20 0.32
TLR8 Q9NR97 4/20 0.31
SLC6A9 P48067 3/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7081102 0.93 GCGR (0.36) GCGRMAOAMAOBNOTUMDHODH
SCHEMBL6974341 0.89
SCHEMBL7087555 0.89 GCGR (0.38) GCGRMAOAMAOBNOTUMDHODH
SCHEMBL6961144 0.87 GCGR (0.39) GCGRMAOAMAOBNOTUMDHODH
SCHEMBL6960474 0.87 TLR8 (0.42) MAOAMAOBNOTUMTLR8NPSR1
SCHEMBL6968511 0.86 MAOA (0.36) GCGRMAOAMAOBNOTUMHAO1
SCHEMBL7084560 0.86 SMN1; SMN2 (0.39) GCGRTLR8
SCHEMBL6967278 0.85 HDAC6 (0.41) MAOAMAOBNOTUMSLC6A9
SCHEMBL7084556 0.84 EPHX1 (0.34) GCGRMAOAMAOBNOTUMSLC6A9
SCHEMBL6970136 0.84 MAOA (0.34) GCGRMAOAMAOBNOTUMDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed