SCHEMBL7084175

SCHEMBL7084175

O=C(O)C1CCN(c2cc(N3CCN(Cc4ccc(C(F)(F)F)cc4C(F)(F)F)CC3)c([N+](=O)[O-])cc2C(F)(F)F)CC1

nearest known ligand 0.77

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 12/20 0.77
CYP2C9 P11712 2/20 0.52
CYP2C19 P33261 2/20 0.52
MAPT P10636 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
POLB P06746 1/20 0.51
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
KMT2A Q03164 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
FFAR2 O15552 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084109 0.89 SERPINE1 (0.82) SERPINE1CYP2C9CYP2C19MAPTCYP1A2
SCHEMBL7165057 0.87 SERPINE1 (1.00) SERPINE1CYP2C9CYP2C19MAPTCYP1A2
SCHEMBL7088169 0.84 SERPINE1 (1.00) SERPINE1CYP2C9CYP2C19MAPTCYP1A2
SCHEMBL7091396 0.82 SERPINE1 (1.00) SERPINE1MAPT
SCHEMBL7084123 0.81 SERPINE1 (0.82) SERPINE1CYP2C9CYP2C19MAPTCYP1A2
SCHEMBL7084622 0.80 SERPINE1 (1.00) SERPINE1CYP2C9CYP2C19MAPTCYP1A2
SCHEMBL29788183 0.79 MAPT (0.80) SERPINE1CYP2C9CYP2C19MAPTCYP1A2
SCHEMBL2039548 0.79 MAPT (0.80) SERPINE1CYP2C9CYP2C19MAPTCYP1A2
SCHEMBL7089079 0.77 SERPINE1 (0.74) SERPINE1CYP2C9CYP2C19MAPTCYP1A2
SCHEMBL7087964 0.77 SERPINE1 (1.00) SERPINE1CYP2C9CYP2C19MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003080060-A1 SUBSTITUTED PIPERAZINE ANTITHROMBOTIC PAI-1 INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 2003-10-02 WO disclosed