SCHEMBL7084201

SCHEMBL7084201

COc1ccc(N(CCCc2cncn2Cc2ccc(C#N)cc2)C(=S)N(Cc2ccccc2C(F)(F)F)OC(=O)CC(O)(CC(=O)O)C(=O)O)cn1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.39
CYP11B2 P19099 3/20 0.39
FNTA P49354 10/20 0.35
FNTB P49356 10/20 0.35
PGGT1B P53609 8/20 0.35
KCNH2 Q12809 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7080524 0.90 CYP11B1 (0.42) CYP11B1CYP11B2FNTAFNTBPGGT1B
SCHEMBL7077080 0.89 CYP11B1 (0.40) CYP11B1CYP11B2FNTAFNTBPGGT1B
Citric Acid SCHEMBL7084194 0.88 CYP11B1 (0.41) CYP11B1CYP11B2FNTAFNTBPGGT1B
SCHEMBL7077584 0.85 CYP11B1 (0.39) CYP11B1CYP11B2FNTAFNTBPGGT1B
Citric Acid SCHEMBL7084202 0.85 CYP11B1 (0.40) CYP11B1CYP11B2FNTAFNTBPGGT1B
Oxalic Acid SCHEMBL7080520 0.81 CYP11B1 (0.46) CYP11B1CYP11B2FNTAFNTBPGGT1B
Cadaverine Tartrate SCHEMBL7077575 0.80 CYP11B1 (0.42) CYP11B1CYP11B2FNTAFNTBPGGT1B
SCHEMBL7168855 0.80 CYP11B1 (0.43) CYP11B1CYP11B2FNTAFNTBPGGT1B
Maleic Acid SCHEMBL7077075 0.80 CYP11B1 (0.42) CYP11B1CYP11B2FNTAFNTBPGGT1B
Oxalic Acid SCHEMBL7080525 0.78 CYP11B1 (0.45) CYP11B1CYP11B2FNTAFNTBPGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1200430-A4 THIOUREA AND ISOTHIOUREA DERIVATIVES FOR INHIBITING RAS-TRANSFORMED CELL GROWTH YUHAN CORP LTD (KR) 2003-01-22 EP disclosed
EP-1200430-A1 THIOUREA AND ISOTHIOUREA DERIVATIVES FOR INHIBITING RAS-TRANSFORMED CELL GROWTH YUHAN CORPORATION, LTD. (KR) 2002-05-02 EP disclosed
WO-2001009128-A1 THIOUREA AND ISOTHIOUREA DERIVATIVES FOR INHIBITING RAS-TRANSFORMED CELL GROWTH YUHAN CORPORATION (KR) 2001-02-08 WO disclosed