SCHEMBL7084316

SCHEMBL7084316

CC(=O)OCC(=O)N1CC=C(c2c(F)cc(N3C[C@H](COc4nc(C)no4)OC3=O)cc2F)CC1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOA P21397 10/20 0.35
GRM2 Q14416 2/20 0.33
BTK Q06187 1/20 0.33
MAOB P27338 5/20 0.32
CALML3 P27482 2/20 0.32
LMNA P02545 1/20 0.32
PTGS1 P23219 1/20 0.32
SDHA P31040 1/20 0.32
F10 P00742 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7078359 0.85 MAOA (0.35) MAOAGRM2BTKMAOBCALML3
SCHEMBL7077034 0.83 MAOA (0.34) MAOAGRM2BTKMAOBCALML3
SCHEMBL7030515 0.81 MAOA (0.51) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL8517728 0.81 MAOA (0.51) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL7081634 0.80 GRM2 (0.36) MAOAGRM2
SCHEMBL7081042 0.80 GRM2 (0.41) GRM2LMNASIGMAR1
SCHEMBL4021263 0.80 MAOA (0.52) MAOAMAOBSIGMAR1
SCHEMBL5237085 0.79 MAOA (0.50) MAOAMAOB
SCHEMBL5833710 0.79 MAOA (0.49) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL7210278 0.77 MAOA (0.44) MAOAMAOBCALML3CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030144263-A1 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them SYNGENTA LIMITED (GB) 2003-07-31 US disclosed
EP-1082323-A2 OXAZOLIDINONE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AstraZeneca UK Limited (GB) 2001-03-14 EP disclosed
WO-1999064417-A2 OXAZOLIDINONE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ASTRAZENECA AB (SE) 1999-12-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030144263-A1 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them CYP3A5, CYP2D6, OXA1L MAOA 1654/4885GRM2 3844/4885BTK 2028/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.