SCHEMBL7085340

SCHEMBL7085340

Nc1nc(N[C@H](CO)Cc2ccccc2)nc2[nH]cnc12

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.47
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
ADORA3 P0DMS8 6/20 0.45
CDK1 P06493 3/20 0.44
CDK5 Q00535 2/20 0.44
ADORA2B P29275 3/20 0.43
ADORA1 P30542 3/20 0.43
MME P08473 1/20 0.42
JAK3 P52333 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
CDK2 P24941 2/20 0.39
CCNE2 O96020 1/20 0.39
CCNE1 P24864 1/20 0.39
CCNA2 P20248 1/20 0.36
CCNA1 P78396 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27564857 1.00 ADORA2A (0.47) ADORA2AKDM4EMEN1MAPTKMT2A
Hydrochloric Acid SCHEMBL7088885 0.99 ADORA2A (0.47) ADORA2AKDM4EMEN1MAPTKMT2A
SCHEMBL13729103 0.77 APP (0.54) ADORA2AMAPTADORA3CDK1ADORA2B
SCHEMBL7658491 0.75 KDM4E (0.44) KDM4EMEN1MAPTKMT2ACDK1
SCHEMBL27763565 0.74 KDM4E (0.43) KDM4EMEN1MAPTKMT2ACDK1
SCHEMBL27763566 0.74 KDM4E (0.43) KDM4EMEN1MAPTKMT2ACDK1
SCHEMBL9792866 0.74 APP (0.57) ADORA2AKMT2AADORA3ADORA2BADORA1
SCHEMBL24669720 0.73 CDK2 (0.65) CDK1CDK5CDK2CCNE2CCNE1
SCHEMBL27763562 0.73 KDM4E (0.42) KDM4EMEN1MAPTKMT2ACDK1
SCHEMBL17815577 0.72 ADORA1 (0.55) ADORA2AADORA3ADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090022-B1 2-(PURIN-9-YL)-TETRAHYDROFURAN-3,4-DIOL DERIVATIVES GLAXO GROUP LTD (GB) 2003-08-06 EP disclosed
US-6495528-B1 ANTIINFLAMMATORY AGENTS; INHIBITING LEUKOCYTE RECRUITMENT AND ACTIVATION; AGONISTS OF ADENOSINE 2A RECEPTOR SMITHKLINE BEECHAM CORPORATION 2002-12-17 US disclosed
CN-1313861-A 2-(purin-9-YL)-tetrahydrofuran-3,4-diolderivatives GLAXO GROUP LTD (GB) 2001-09-19 CN disclosed