SCHEMBL7086341

SCHEMBL7086341

Nc1ccc2c(c1)C(=C(Nc1cccnc1)c1ccccc1)C(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.44
ALDH1A1 P00352 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PDPK1 O15530 3/20 0.41
AKT2 P31751 1/20 0.41
TGM2 P21980 4/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PKM P14618 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 2/20 0.40
HIF1A Q16665 1/20 0.40
KMT2A Q03164 1/20 0.39
GAA P10253 1/20 0.39
KCNK3 O14649 1/20 0.39
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7086337 1.00 NAMPT (0.44) NAMPTALDH1A1L3MBTL1PDPK1AKT2
SCHEMBL7086762 0.89 PDPK1 (0.45) PDPK1AKT2
SCHEMBL29643001 0.89 PDPK1 (0.45) PDPK1AKT2
SCHEMBL7086761 0.89 PDPK1 (0.45) PDPK1AKT2
SCHEMBL7086305 0.88 BACE1 (0.45) PDPK1AKT2
SCHEMBL7086310 0.88 BACE1 (0.45) PDPK1AKT2
SCHEMBL7239292 0.86 PDPK1 (0.43) NAMPTALDH1A1PDPK1AKT2TGM2
SCHEMBL7239288 0.86 PDPK1 (0.43) NAMPTALDH1A1PDPK1AKT2TGM2
SCHEMBL7087980 0.85 PDPK1 (0.50) ALDH1A1PDPK1AKT2SMN1; SMN2LMNA
SCHEMBL7087977 0.85 PDPK1 (0.50) ALDH1A1PDPK1AKT2SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071665-B1 SUBSTITUTED INDOLINONES HAVING AN INHIBITING EFFECT ON KINASES AND CYCLINE/CDK COMPLEXES BOEHRINGER INGELHEIM PHARMA (DE) 2003-10-01 EP disclosed
US-6169106-B1 ANTITUMOUR AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-01-02 US disclosed