SCHEMBL7086384

SCHEMBL7086384

CCOP(=O)(OCC)C(Cc1cc(C)c(O)c(C(C)(C)C)c1)P(=O)(OCC)OCC

nearest known ligand 0.85

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 13/20 0.85
NR1I2 O75469 1/20 0.44
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
GAA P10253 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
PKM P14618 1/20 0.36
HTT P42858 1/20 0.36
HSPA5 P11021 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704691 0.92 HMGCR (1.00) HMGCRNR1I2CYP1A2CYP2C9CYP2C19
SCHEMBL7086181 0.84 HMGCR (0.85) HMGCR
SCHEMBL9723401 0.82 HMGCR (0.81) HMGCRNR1I2CYP1A2CYP2C9CYP2C19
SCHEMBL7526269 0.82 HMGCR (0.56) HMGCRCYP1A2CYP2C9CYP2C19GAA
SCHEMBL7083916 0.81 HMGCR (0.80) HMGCRNR1I2CYP1A2CYP2C9CYP2C19
SCHEMBL7134552 0.79 HMGCR (0.76) HMGCRNR1I2CYP1A2GAAMEN1
SCHEMBL15705739 0.78 HMGCR (0.52) HMGCRNR1I2CYP1A2CYP2C9CYP2C19
SCHEMBL7084466 0.77 HMGCR (0.74) HMGCRNR1I2CYP1A2CYP2C9CYP2C19
SCHEMBL9723334 0.76 HMGCR (0.71) HMGCRNR1I2CYP1A2CYP2C9CYP2C19
Apomine SCHEMBL1648488 0.75 HMGCR (1.00) HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326618-A2 USE OF ARYL-SUBSTITUTED 1,1-DIPHOSPHONATES FOR THE TREATMENT OF BONE DISEASES Ilex Oncology Research S.A. (CH) 2003-07-16 EP claimed
WO-2002011704-A2 USE OF ARYL-SUBSTITUTED 1,1-DIPHOSPHONATES FOR THE TREATMENT OF BONE DISEASES SYMPHAR S.A. (CH) 2002-02-14 WO claimed
EP-0845991-B1 USE OF PHENOL SUBSTITUTED DIPHOSPHONATES AS ANTINEOPLASTIC AGENTS SYMPHAR SA (CH) 2002-02-06 EP claimed
US-6127350-A FOR TREATMENT AND PREVENTION OF RAS ONCOGENE DEPENDENT CANCERS AND METASTATIC INVASIONS SYMPHAR S.A. (SE) 2000-10-03 US claimed
US-5043330-A Antiinflammatory and hypotensive agents; antihyperlipemia SYMPHAR S.A. (CH) 1991-08-27 US claimed
US-5128331-A Gen-diphosphonates SYMPHAR S.A. (CH) 1992-07-07 US disclosed