SCHEMBL7086568

SCHEMBL7086568

CO/N=C1\C[C@@H](C(=O)NC[C@@H](O)c2ccccc2)N(C(=O)c2ccc(-c3c(C)cccc3C)cc2)C1

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OXTR P30559 5/20 0.85
AVPR1A P37288 3/20 0.85
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35
MMP1 P03956 1/20 0.35
MMP3 P08254 1/20 0.35
MMP7 P09237 1/20 0.35
CFD P00746 1/20 0.34
BCAT2 O15382 1/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
ROCK2 O75116 2/20 0.34
ROCK1 Q13464 2/20 0.34
MEN1 O00255 1/20 0.34
PABPC1 P11940 1/20 0.34
KMT2A Q03164 1/20 0.34
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7086784 0.94 OXTR (0.74) OXTRAVPR1ALMNAPKMMMP1
SCHEMBL5478502 0.92 OXTR (0.72) OXTRAVPR1ALMNAKDM4EMEN1
SCHEMBL5478504 0.92 OXTR (0.72) OXTRAVPR1ALMNAKDM4EMEN1
SCHEMBL4936354 0.92 OXTR (1.00) OXTRAVPR1ALMNAPKMMMP1
SCHEMBL4936174 0.92 OXTR (1.00) OXTRAVPR1ALMNAPKMMMP1
SCHEMBL5743785 0.92 OXTR (1.00) OXTRAVPR1ALMNAPKMMMP1
SCHEMBL4943198 0.92 OXTR (1.00) OXTRAVPR1ALMNAPKMMMP1
SCHEMBL4942975 0.92 OXTR (1.00) OXTRAVPR1ALMNAPKMMMP1
SCHEMBL5743780 0.92 OXTR (1.00) OXTRAVPR1ALMNAPKMMMP1
SCHEMBL4940385 0.92 OXTR (1.00) OXTRAVPR1ALMNAPKMMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268419-A1 PYRROLIDINE DERIVATIVES USEFUL AS BAX INHIBITORS Applied Research Systems ARS Holding N.V. (AN) 2003-01-02 EP disclosed
WO-2001072705-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-04 WO disclosed