SCHEMBL7086602

SCHEMBL7086602

CCn1c(COC(=O)NC)nc(C(C)C)c1Sc1cccc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.34
TOP2B Q02880 1/20 0.34
DHODH Q02127 1/20 0.34
ENPP2 Q13822 1/20 0.34
SLC6A9 P48067 5/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 1/20 0.32
MAOB P27338 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
EPHX1 P07099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974435 0.90 TOP2A (0.32) TOP2ATOP2BENPP2
SCHEMBL6974491 0.89 MEN1 (0.37) DHODHSLC6A9CA2CA4ALDH1A1
SCHEMBL7078929 0.89 TP53 (0.37) TOP2ATOP2BSLC6A9ALDH1A1LMNA
SCHEMBL6969443 0.89 DHODH (0.32) DHODH
SCHEMBL6974432 0.89 EPHX1 (0.35) DHODHSLC6A9CA2CA4ALDH1A1
SCHEMBL6969410 0.89 TOP2A (0.35) TOP2ATOP2BENPP2SLC6A9CA2
SCHEMBL7087523 0.88 TOP2A (0.44) TOP2ATOP2BALDH1A1LMNAMAPT
SCHEMBL6967603 0.88 ENPP2 (0.40) TOP2ATOP2BENPP2LMNAMAPT
SCHEMBL7081406 0.86 IRAK4 (0.37) ALDH1A1LMNAMAPTCYP1A2CYP3A4
SCHEMBL7081110 0.86 S1PR3 (0.39) ENPP2SLC6A9LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed