SCHEMBL7086637

SCHEMBL7086637

CO/N=C1\C[C@@H](C(=O)NCCCCO)N(C(=O)c2ccc(-c3ccccc3)cc2)C1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OXTR P30559 5/20 0.70
AVPR1A P37288 3/20 0.61
LMNA P02545 2/20 0.43
TLR2 O60603 4/20 0.39
TLR1 Q15399 4/20 0.39
DRD2 P14416 3/20 0.38
DRD3 P35462 3/20 0.38
MMP1 P03956 1/20 0.38
MMP3 P08254 1/20 0.38
MMP7 P09237 1/20 0.38
DRD4 P21917 1/20 0.38
KCNH2 Q12809 1/20 0.38
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4942292 1.00 OXTR (0.70) OXTRAVPR1ALMNATLR2TLR1
SCHEMBL4942110 0.97 OXTR (0.71) OXTRAVPR1ALMNATLR2TLR1
SCHEMBL4939162 0.93 OXTR (0.73) OXTRAVPR1ALMNAMMP1MMP3
SCHEMBL4944329 0.93 OXTR (0.73) OXTRAVPR1ALMNAMMP1MMP3
SCHEMBL4943696 0.89 OXTR (0.72) OXTRAVPR1ALMNAMMP1MMP3
SCHEMBL7086396 0.88 AVPR1A (0.73) OXTRAVPR1ALMNADRD2DRD3
SCHEMBL4940423 0.88 AVPR1A (0.73) OXTRAVPR1ALMNADRD2DRD3
SCHEMBL7088615 0.87 OXTR (0.70) OXTRAVPR1ALMNATLR2TLR1
SCHEMBL7164251 0.87 OXTR (0.70) OXTRAVPR1ALMNAMMP1MMP3
SCHEMBL4943384 0.87 OXTR (0.70) OXTRAVPR1ALMNATLR2TLR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268418-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS Applied Research Systems ARS Holding N.V. (AN) 2003-01-02 EP disclosed
WO-2001074769-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-11 WO disclosed