SCHEMBL7089907

SCHEMBL7089907

Cc1cccc(Nc2n[nH]c(Sc3ccsc3)n2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 2/20 0.43
CDK2 P24941 2/20 0.42
SRC P12931 1/20 0.42
ZAP70 P43403 1/20 0.42
SYK P43405 1/20 0.42
AURKA O14965 1/20 0.41
GAA P10253 1/20 0.40
SLC2A1 P11166 1/20 0.39
GRM4 Q14833 1/20 0.39
CCR4 P51679 1/20 0.39
CDK1 P06493 2/20 0.39
CCNB1 P14635 2/20 0.39
CCNA2 P20248 1/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
HTT P42858 2/20 0.38
KCNH3 Q9ULD8 1/20 0.38
MEN1 O00255 3/20 0.38
RAB9A P51151 3/20 0.38
KMT2A Q03164 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7088181 0.85 GAA (0.48) NFKB1CDK2AURKAGAACDK1
SCHEMBL5385474 0.82 NFKB1 (0.40) NFKB1CDK2SRCZAP70SYK
SCHEMBL7089497 0.80 PIK3CA (0.42) NFKB1CDK2SRCZAP70SYK
SCHEMBL6983370 0.80 NFKB1 (0.42) NFKB1CDK2SRCZAP70SYK
SCHEMBL7087580 0.80 CDK2 (0.46) NFKB1CDK2SRCZAP70SYK
SCHEMBL7087411 0.80 NFKB1 (0.44) NFKB1CDK2SRCZAP70SYK
SCHEMBL7090453 0.78 NFKB1 (0.46) NFKB1CDK2SRCZAP70SYK
SCHEMBL7088195 0.78 NFKB1 (0.48) NFKB1CDK2SRCZAP70SYK
SCHEMBL7083578 0.78 NPC1 (0.38) CDK2SYKAURKAKCNH3MEN1
SCHEMBL7087516 0.77 NFKB1 (0.44) NFKB1CDK2SRCZAP70SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1223932-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2003-01-15 EP disclosed
EP-1223932-A1 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2002-07-24 EP disclosed
WO-2001024796-A1 1,2,4-TRIAZOLE DERIVATIVES, COMPOSITION, PROCESS OF MAKING AND METHODS OF USE SMITHKLINE BEECHAM CORPORATION (US) 2001-04-12 WO disclosed