SCHEMBL7090697

SCHEMBL7090697

NS(=O)(=O)c1ccc(C2NC(=O)NC2c2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 15/20 0.50
CA9 Q16790 15/20 0.50
CA1 P00915 14/20 0.50
CA12 O43570 13/20 0.50
CA7 P43166 8/20 0.50
CA14 Q9ULX7 3/20 0.50
CA3 P07451 1/20 0.50
CA4 P22748 1/20 0.50
CA6 P23280 1/20 0.50
CA5A P35218 1/20 0.50
PLA2G7 Q13093 1/20 0.50
CA13 Q8N1Q1 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
PTGS2 P35354 3/20 0.46
SOS1 Q07889 1/20 0.44
KDM1A O60341 1/20 0.41
MAOA P21397 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2724029 0.81 SMN1; SMN2 (0.52) CA2
SCHEMBL2724030 0.81 SMN1; SMN2 (0.52) CA2
SCHEMBL15669988 0.70 SMN1; SMN2 (0.54) CA2
Benzenesulfonamide SCHEMBL28257999 0.70 CA2 (1.00) CA2CA9CA1CA12CA7
Benzenesulfonamide SCHEMBL729 0.70 CA2 (1.00) CA2CA9CA1CA12CA7
Benzenesulfonamide SCHEMBL29825137 0.70 CA2 (1.00) CA2CA9CA1CA12CA7
SCHEMBL19479299 0.70 CA2 (1.00) CA2CA9CA1CA12CA7
Benzenesulfonamide SCHEMBL1332409 0.70 CA2 (1.00) CA2CA9CA1CA12CA7
Benzenesulfonamide SCHEMBL6868390 0.70 CA2 (1.00) CA2CA9CA1CA12CA7
SCHEMBL9741405 0.69 CYP19A1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030050330-A1 4,5-subtstituted imdazolyl compounds for the treatment of inflammation G.D. SEARLE & CO. 2003-03-13 US disclosed
EP-0772601-B1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2002-09-18 EP disclosed
US-6426360-B1 ANTIARTHRITIC AGENTS G D SEARLE & CO. 2002-07-30 US disclosed
EP-1211244-A2 4,5-substitued imidazolyl compounds for the treatment of inflammation G.D. Searle & Co. (US) 2002-06-05 EP disclosed
US-5620999-A ANTIARTHRITIC, ANALGESIC AND ANTIPYRATIC AGENT G.D. SEARLE & CO. 1997-04-15 US disclosed
WO-1996003387-A1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030050330-A1 4,5-subtstituted imdazolyl compounds for the treatment of inflammation AHR, HACL2, IRAK2 CA2 3267/4885CA9 2915/4885CA1 4768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.