SCHEMBL7091805

SCHEMBL7091805

CCCOc1cc2c(cc1C(=O)OC)CC(N(CCC)CCC)C2

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.57
CYP2D6 P10635 1/20 0.57
CYP2C9 P11712 1/20 0.57
ALOX15 P16050 1/20 0.57
MAPK1 P28482 1/20 0.57
FYN P06241 1/20 0.49
DRD3 P35462 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7093200 0.95 ALDH1A1 (0.57) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1
SCHEMBL7093657 0.91 ALDH1A1 (0.58) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1
SCHEMBL8688816 0.89 ALDH1A1 (0.69) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1
SCHEMBL7447619 0.87 ALDH1A1 (0.60) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1
SCHEMBL7093125 0.86 ALDH1A1 (0.55) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1
SCHEMBL8442018 0.85 ALDH1A1 (0.57) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1
SCHEMBL7090289 0.84 ALDH1A1 (0.53) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1
SCHEMBL7092974 0.82 FYN (0.66) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1
SCHEMBL7092696 0.82 ALDH1A1 (0.52) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1
SCHEMBL27515209 0.80 ALDH1A1 (0.56) ALDH1A1CYP2D6CYP2C9ALOX15MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923542-B1 ARYL SUBSTITUTED CYCLIC AMINES AS SELECTIVE DOPAMINE D3 LIGANDS UPJOHN CO (US) 2003-08-20 EP disclosed
US-6084130-A FOR TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS PHARMACIA & UPJOHN COMPANY (US) 2000-07-04 US disclosed
EP-0923542-A1 ARYL SUBSTITUTED CYCLIC AMINES AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1999-06-23 EP disclosed
WO-1997045403-A1 ARYL SUBSTITUTED CYCLIC AMINES AS SELECTIVE DOPAMINE D3 LIGANDS PHARMACIA & UPJOHN COMPANY (US) 1997-12-04 WO disclosed