SCHEMBL7091944

SCHEMBL7091944

COc1cccc(-c2nc(Nc3ccc4[nH]ncc4c3)c3c(F)cccc3n2)c1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 12/20 0.62
ROCK1 Q13464 6/20 0.55
CLK2 P49760 1/20 0.54
BLK P51451 1/20 0.54
CSNK2A1 P68400 1/20 0.54
STK3 Q13188 1/20 0.54
DYRK1A Q13627 1/20 0.54
AURKB Q96GD4 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
STK17A Q9UEE5 1/20 0.54
ABCG2 Q9UNQ0 5/20 0.53
ABCB1 P08183 2/20 0.52
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
KDR P35968 1/20 0.48
SYK P43405 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3578405 0.93 ROCK2 (0.63) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL5737426 0.88 ROCK2 (0.55) ROCK2ROCK1CLK2BLKCSNK2A1
Hydrochloric Acid SCHEMBL3585306 0.87 ROCK2 (0.54) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL3590236 0.86 ROCK2 (0.78) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL5737623 0.86 ROCK2 (0.53) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL3589828 0.86 ROCK2 (0.53) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL3588269 0.85 MKNK1 (0.54) ROCK2ROCK1CLK2BLKCSNK2A1
Hydrochloric Acid SCHEMBL3580794 0.85 ROCK2 (0.52) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL3583259 0.83 ROCK2 (0.64) ROCK2ROCK1CLK2BLKCSNK2A1
SCHEMBL3589238 0.83 ROCK2 (0.49) ROCK2ROCK1CLK2BLKCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1370553-A2 RHO-KINASE INHIBITORS Bayer Corporation (US) 2003-12-17 EP disclosed
WO-2002076976-A2 RHO-KINASE INHIBITORS BAYER CORPORATION (US) 2002-10-03 WO disclosed