SCHEMBL7093764

SCHEMBL7093764

Cc1cccc(Cn2nc(-c3ccco3)c3cnc(N)nc32)c1

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.73
ADORA1 P30542 19/20 0.73
ADORA3 P0DMS8 3/20 0.62
ADORA2B P29275 3/20 0.62
HDAC1 Q13547 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4455442 0.84 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL4044853 0.76 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3269171 0.76 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL4219305 0.76 ADORA2A (0.49) ADORA2AADORA1ADORA2B
SCHEMBL4452802 0.74 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL13601224 0.72 ADORA2A (0.81) ADORA2AADORA1HDAC1
SCHEMBL4452849 0.72 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL4449511 0.72 ADORA2A (0.76) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL4456961 0.72 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2BHDAC1
SCHEMBL20118706 0.72 ADORA1 (0.56) ADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349552-A1 PYRAZOLO 3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055082-A1 PYRAZOLO[3,4-D]PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed