SCHEMBL7096088

SCHEMBL7096088

C[C@]12CCC3c4ccc(NS(=O)(=O)O)cc4CCC3C1C[C@@H](O)[C@@H]2O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.68
ESR2 Q92731 4/20 0.68
LMNA P02545 3/20 0.68
CYP2C9 P11712 2/20 0.68
CYP2C19 P33261 2/20 0.68
HIF1A Q16665 2/20 0.68
NR3C1 P04150 2/20 0.68
SHBG P04278 2/20 0.68
PGR P06401 2/20 0.68
SERPINA6 P08185 2/20 0.68
AR P10275 2/20 0.68
SLC6A4 P31645 2/20 0.68
SNCA P37840 2/20 0.68
SLC6A3 Q01959 2/20 0.68
PTGS1 P23219 1/20 0.68
OR51E2 Q9H255 1/20 0.68
UGT1A10 Q9HAW8 1/20 0.68
MAPT P10636 2/20 0.58
USP2 O75604 1/20 0.58
MAPK1 P28482 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3908652 0.87 ABCC1 (0.70) ESR1ESR2LMNACYP2C9CYP2C19
Estriol SCHEMBL10412523 0.85 ESR1 (0.89) ESR1ESR2LMNACYP2C9CYP2C19
Estriol SCHEMBL6438208 0.85 ESR1 (0.89) ESR1ESR2LMNACYP2C9CYP2C19
SCHEMBL17515286 0.85 ABCC4 (0.56) ESR1ESR2LMNACYP2C9CYP2C19
Estriol SCHEMBL7992695 0.84 ESR1 (0.87) ESR1ESR2LMNACYP2C9CYP2C19
SCHEMBL17515288 0.84 ABCC1 (0.58) ESR1ESR2LMNACYP2C9CYP2C19
Estriol SCHEMBL345572 0.83 ESR1 (0.85) ESR1ESR2LMNACYP2C9CYP2C19
SCHEMBL17515287 0.83 ABCC4 (0.52) ESR1ESR2LMNACYP2C9CYP2C19
SCHEMBL5521870 0.82 ABCC4 (0.76) ESR1ESR2LMNACYP2C9CYP2C19
SCHEMBL2517551 0.82 ABCC4 (0.76) ESR1ESR2LMNACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775156-B1 PHARMACEUTICAL COMPOSITIONS CONTAINING ESTRA-1,3,5(10)-TRIENE DERIVATIVES JENAPHARM GMBH (DE) 2003-09-03 EP claimed