SCHEMBL7100486

SCHEMBL7100486

Cc1ccnc(NCCCCC(=O)NC(=O)NNC(CC(=O)O)c2ccccc2)c1

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.62
ITGB3 P05106 19/20 0.62
ITGB6 P18564 8/20 0.62
ITGB5 P18084 7/20 0.62
ITGA2B P08514 6/20 0.61
ITGB1 P05556 1/20 0.49
ITGA5 P08648 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7105210 0.92 ITGAV (0.59) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7104969 0.92 ITGAV (0.66) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7099706 0.90 ITGAV (0.77) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7099672 0.89 ITGAV (0.78) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7103817 0.88 ITGAV (0.61) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7104917 0.87 ITGAV (0.61) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7102208 0.86 ITGAV (0.58) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7104922 0.81 ITGB3 (0.89) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL6670827 0.78 ITGAV (0.79) ITGAVITGB3ITGB6ITGB5ITGA2B
SCHEMBL7172749 0.77 ITGAV (0.77) ITGAVITGB3ITGB6ITGB5ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed