SCHEMBL710057

SCHEMBL710057

Cc1cc(Nc2ccc(S(=O)(=O)Nc3nccs3)cc2)n(-c2ccc(Cl)cc2)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.60
LMNA P02545 2/20 0.60
SCN9A Q15858 6/20 0.56
PPIA P62937 3/20 0.55
GAA P10253 2/20 0.54
HPGD P15428 1/20 0.54
MAPT P10636 1/20 0.52
ALPG P10696 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CCNT1 O60563 1/20 0.51
CDK9 P50750 1/20 0.51
AVPR2 P30518 1/20 0.50
GPR27 Q9NS67 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
PTGS2 P35354 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
SCN3A Q9NY46 1/20 0.49
ALOX12 P18054 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL712299 0.90 SCN9A (0.68) SMN1; SMN2SCN9AGAAHPGDCA1
SCHEMBL712100 0.86 SCN9A (0.63) SMN1; SMN2LMNASCN9AGAAHPGD
SCHEMBL714461 0.85 LMNA (0.57) SMN1; SMN2LMNASCN9APPIACCNT1
SCHEMBL712049 0.80 SCN9A (0.54) SMN1; SMN2LMNASCN9AGAAHPGD
SCHEMBL712667 0.79 SCN9A (0.65) SCN9APPIAMAPTNPSR1MEN1
SCHEMBL714318 0.79 SCN9A (0.65) SCN9AMEN1KMT2A
SCHEMBL713724 0.78 NAMPT (0.52) SMN1; SMN2LMNASCN9APPIAMEN1
SCHEMBL710624 0.78 SCN9A (0.55) SMN1; SMN2LMNASCN9AGAAHPGD
SCHEMBL712390 0.78 SCN9A (0.55) SMN1; SMN2LMNASCN9AGAAHPGD
Sulfazamet SCHEMBL28264721 0.78 SCN9A (0.67) SMN1; SMN2LMNASCN9AMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8124610-B2 Sodium channel inhibitors ICAGEN INC. (US) 2012-02-28 US claimed
US-8124610-B2 Sodium channel inhibitors ICAGEN INC. (US) 2012-02-28 US disclosed
EP-2173743-A2 SODIUM CHANNEL INHIBITORS Icagen, Inc. (US) 2010-04-14 EP disclosed
US-20090023740-A1 SODIUM CHANNEL INHIBITORS ICAGEN (US) 2009-01-22 US disclosed
WO-2009012242-A2 SODIUM CHANNEL INHIBITORS ICAGEN, INC. (US) 2009-01-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090023740-A1 SODIUM CHANNEL INHIBITORS TRPV1, SCN1A, SCN2A SMN1; SMN2 287/4885LMNA 2921/4885SCN9A 17/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.