Benzothiophene

Benzothiophene

SCHEMBL7101018

OCc1cc2ccccc2s1.c1ccc2sccc2c1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.77
ASIC3 Q9UHC3 1/20 0.51
LOXL2 Q9Y4K0 1/20 0.51
AGXT P21549 1/20 0.47
ADRB2 P07550 1/20 0.47
CTNNB1 P35222 1/20 0.41
WNT3A P56704 1/20 0.41
ADRA1D P25100 2/20 0.40
MGLL Q99685 1/20 0.40
IDH1 O75874 1/20 0.39
BCL2L1 Q07817 1/20 0.39
SLC5A2 P31639 3/20 0.38
APP P05067 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL355949 0.88 CYP2A6 (1.00) CYP2A6ASIC3LOXL2AGXTADRB2
Benzothiophene SCHEMBL6151566 0.76 CTNNB1 (0.41) CYP2A6ADRB2CTNNB1WNT3A
Benzothiophene SCHEMBL4378682 0.75 CTNNB1 (0.46) CYP2A6CTNNB1WNT3AMGLLBCL2L1
Benzothiophene SCHEMBL28758675 0.75 CTNNB1 (0.46) CYP2A6CTNNB1WNT3AMGLLBCL2L1
Benzothiophene SCHEMBL29415494 0.75
Benzothiophene SCHEMBL28545602 0.75 CA12 (0.42) CYP2A6ASIC3LOXL2CTNNB1WNT3A
Benzothiophene SCHEMBL7023 0.75
Benzothiophene SCHEMBL29383883 0.75
Benzothiophene SCHEMBL451494 0.75
Benzothiophene SCHEMBL253491 0.75 CA12 (0.42) CYP2A6ASIC3LOXL2CTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003101994-A1 FUSED BICYCLIC AROMATIC COMPOUNDS THAT ARE USEFUL IN TREATING SEXUAL DYSFUNCTION ABBOTT LABORATORIES (US) 2003-12-11 WO disclosed