SCHEMBL7101164

SCHEMBL7101164

NC(=O)C12C(=O)CO[C@H]1CCCN2C(=O)[CH]Cc1ccccc1

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
F2 P00734 6/20 0.32
POLB P06746 2/20 0.31
DPP4 P27487 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31
DPP7 Q9UHL4 1/20 0.31
PRSS1 P07477 2/20 0.31
GAA P10253 2/20 0.31
LMNA P02545 1/20 0.31
TSHR P16473 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
ALDH1A1 P00352 2/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4449150 1.00 HCRTR1 (0.32) HCRTR1HCRTR2F2POLBDPP4
SCHEMBL4446611 0.94 F2 (0.32) F2POLBGAALMNATSHR
SCHEMBL7100766 0.94 F2 (0.32) F2POLBGAALMNATSHR
SCHEMBL7101601 0.91 DPP4 (0.31) DPP4
SCHEMBL4448316 0.91 DPP4 (0.31) DPP4
SCHEMBL4450150 0.89 CYP2C19 (0.32) NPC1ALDH1A1
SCHEMBL7102347 0.84
SCHEMBL4448472 0.84
SCHEMBL5092214 0.84
SCHEMBL6803954 0.84 CHRM2 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362052-A1 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES Amura Therapeutics Limited (GB) 2003-11-19 EP disclosed
WO-2002057270-A1 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES AMURA THERAPEUTICS LIMITED (GB) 2002-07-25 WO disclosed