SCHEMBL7102178

SCHEMBL7102178

O=C1OCC2=C1C(c1ccccc1C(F)(F)F)C1=C(COC1=O)N2

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
ABCC9 O60706 7/20 0.47
KCNJ11 Q14654 7/20 0.47
ABCC8 Q09428 6/20 0.47
KCNJ8 Q15842 6/20 0.47
KDM4E B2RXH2 4/20 0.42
LMNA P02545 3/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 2/20 0.42
HPGD P15428 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
GSK3B P49841 3/20 0.42
GSK3A P49840 2/20 0.42
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10817848 0.88 ALDH1A1 (0.46) ALDH1A1ABCC9KCNJ11ABCC8KCNJ8
SCHEMBL7100697 0.87 GSK3B (0.60) ALDH1A1KDM4ELMNAMAPTHPGD
SCHEMBL28969774 0.85 ALDH1A1 (0.41) ALDH1A1ABCC9KCNJ11ABCC8KCNJ8
SCHEMBL28969770 0.85 ALDH1A1 (0.41) ALDH1A1ABCC9KCNJ11ABCC8KCNJ8
SCHEMBL9865585 0.83 CYP1A2 (0.58) ALDH1A1KDM4EMAPTHPGDKMT2A
SCHEMBL7096837 0.82 ALDH1A1 (0.52) ALDH1A1ABCC9KCNJ11ABCC8KCNJ8
SCHEMBL24117078 0.81 CACNA1C (0.48) ALDH1A1KDM4EMAPTHPGDKMT2A
SCHEMBL11003495 0.81 KDM4E (0.69) ALDH1A1KDM4E
SCHEMBL30266638 0.81 CACNA1C (0.48) ALDH1A1KDM4EMAPTHPGDKMT2A
SCHEMBL7099081 0.81 ALDH1A1 (0.66) ALDH1A1ABCC9KCNJ11ABCC8KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1278746-A2 DIHYDROPYRIDINE COMPOUNDS AND METHODS OF USE Abbott Laboratories (US) 2003-01-29 EP claimed
WO-2001083480-A2 DIHYDROPYRIDINE COMPOUNDS AND METHODS OF USE ABBOTT LABORATORIES (US) 2001-11-08 WO claimed
EP-1131322-A2 DIHYDROPYRIDINE COMPOUNDS AND METHODS OF USE ABBOTT LABORATORIES (US) 2001-09-12 EP claimed
WO-2000024741-A2 DIHYDROPYRIDINE COMPOUNDS AND THEIR USE AS POTASSIUM CHANNEL OPENERS ABBOTT LABORATORIES (US) 2000-05-04 WO claimed
EP-1278746-A2 DIHYDROPYRIDINE COMPOUNDS AND METHODS OF USE Abbott Laboratories (US) 2003-01-29 EP disclosed
WO-2001083480-A2 DIHYDROPYRIDINE COMPOUNDS AND METHODS OF USE ABBOTT LABORATORIES (US) 2001-11-08 WO disclosed
EP-1131322-A2 DIHYDROPYRIDINE COMPOUNDS AND METHODS OF USE ABBOTT LABORATORIES (US) 2001-09-12 EP disclosed
WO-2000024741-A2 DIHYDROPYRIDINE COMPOUNDS AND THEIR USE AS POTASSIUM CHANNEL OPENERS ABBOTT LABORATORIES (US) 2000-05-04 WO disclosed