SCHEMBL7102550

SCHEMBL7102550

CNN1CCC[C@H](c2cnc(Br)c(F)c2)C1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 3/20 0.33
HRH2 P25021 1/20 0.32
HRH1 P35367 1/20 0.32
HRH4 Q9H3N8 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
DRD2 P14416 1/20 0.32
DRD1 P21728 1/20 0.32
DRD4 P21917 1/20 0.32
DRD5 P21918 1/20 0.32
DRD3 P35462 1/20 0.32
PDE2A O00408 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7103964 1.00 PROKR1 (0.33) PROKR1HRH2HRH1HRH4HRH3
SCHEMBL7103286 0.96 HRH2 (0.33) PROKR1HRH2HRH1HRH4HRH3
SCHEMBL7103477 0.96 HRH2 (0.33) PROKR1HRH2HRH1HRH4HRH3
SCHEMBL7099165 0.92 PARP1 (0.31) HRH4HRH3
SCHEMBL7492241 0.92 PARP1 (0.31) HRH4HRH3
SCHEMBL7488469 0.90 PARP1 (0.32) HRH2HRH1HRH4HRH3
SCHEMBL7100525 0.90 PARP1 (0.32) HRH2HRH1HRH4HRH3
SCHEMBL7101894 0.85 PROKR1 (0.35) PROKR1HRH2HRH1HRH4HRH3
SCHEMBL7101551 0.85 SLC6A2 (0.36) PROKR1HRH2HRH1HRH4HRH3
SCHEMBL7100533 0.85 SLC6A2 (0.36) PROKR1HRH2HRH1HRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500402-A 2003-01-07 JP claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP claimed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP disclosed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO disclosed