SCHEMBL7103286

SCHEMBL7103286

CNN1CCCC[C@@H](c2cnc(Br)c(F)c2)C1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 1/20 0.33
HRH1 P35367 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
PROKR1 Q8TCW9 5/20 0.32
PDGFRB P09619 1/20 0.31
PDGFRA P16234 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7103477 1.00 HRH2 (0.33) HRH2HRH1HRH4HRH3PROKR1
SCHEMBL7103964 0.96 PROKR1 (0.33) HRH2HRH1HRH4HRH3PROKR1
SCHEMBL7102550 0.96 PROKR1 (0.33) HRH2HRH1HRH4HRH3PROKR1
SCHEMBL7492241 0.91 PARP1 (0.31) HRH4HRH3
SCHEMBL7099165 0.91 PARP1 (0.31) HRH4HRH3
SCHEMBL7488469 0.86 PARP1 (0.32) HRH2HRH1HRH4HRH3PDGFRB
SCHEMBL7100525 0.86 PARP1 (0.32) HRH2HRH1HRH4HRH3PDGFRB
SCHEMBL7102133 0.85 SLC6A2 (0.41) HRH2HRH1HRH4HRH3PROKR1
SCHEMBL7101818 0.85 PROKR1 (0.36) HRH2HRH1HRH4HRH3PROKR1
SCHEMBL7102607 0.85 SLC6A2 (0.41) HRH2HRH1HRH4HRH3PROKR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2003500402-A 2003-01-07 JP claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP claimed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO claimed
EP-1178982-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2002-02-13 EP disclosed
WO-2000071534-A1 HETEROCYCLIC SUBSTITUTED AMINOAZACYCLES USEFUL AS CENTRAL NERVOUS SYSTEM AGENTS ABBOTT LABORATORIES (US) 2000-11-30 WO disclosed