SCHEMBL7103370

SCHEMBL7103370

COc1ccc2ccccc2c1C1CCN(CCn2cnc3sc(C(=O)N(C)C)c(C)c3c2=O)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.48
ADRA1D P25100 1/20 0.48
HTR1B P28222 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
ALDH1A1 P00352 4/20 0.47
THRB P10828 3/20 0.47
HPGD P15428 3/20 0.47
SIRT2 Q8IXJ6 9/20 0.44
KDM4E B2RXH2 4/20 0.43
RXFP1 Q9HBX9 2/20 0.43
PPARG P37231 1/20 0.43
NR2E3 Q9Y5X4 1/20 0.43
NCOR2 Q9Y618 1/20 0.43
P2RX3 P56373 3/20 0.43
GAA P10253 2/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7014582 0.87 HTR1A (0.65) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7012836 0.86 KDM4E (0.49) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7005853 0.86 HTR1A (0.45) HTR1AADRA1DHTR1BADRA1AADRA1B
Water SCHEMBL7720208 0.86 HTR1A (0.64) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7012662 0.80 HTR1A (0.52) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7013844 0.80 HTR1A (0.62) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7012872 0.80 HTR1A (0.62) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7013973 0.77 HTR1A (0.58) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7014939 0.76 HTR1A (0.63) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7013768 0.76 HTR1A (0.62) HTR1AADRA1DHTR1BADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0988306-B1 3-SUBSTITUTED 3,4 DIHYDRO-THIENO 2, 3-D]PYRIMIDINE DERIVATIVES AND PRODUCTION AND USE OF THE SAME ABBOTT GMBH & CO KG (DE) 2003-07-09 EP disclosed
US-6387912-B1 STROKE THERAPY BASF AKTIENGESELLSCHAFT (DE) 2002-05-14 US disclosed
US-6159962-A 3-substituted 3,4-dihydro-thieno[2,3-D]pyrimidine derivatives and production and use of the same BASF AKTIENGESELLSCHAFT (DE) 2000-12-12 US disclosed