SCHEMBL7103716

SCHEMBL7103716

O=C(O)CCCC(=O)NNC(=O)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.68
EPHX2 P34913 1/20 0.51
CASP3 P42574 2/20 0.46
FABP5 Q01469 3/20 0.44
FABP7 O15540 2/20 0.44
MDM4 O15151 1/20 0.41
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.40
MEN1 O00255 1/20 0.40
ALPL P05186 1/20 0.40
ALPI P09923 1/20 0.40
ALPG P10696 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13878698 0.88 KMT2A (0.65) KMT2AEPHX2CASP3FABP5FABP7
SCHEMBL5557575 0.85 KMT2A (0.73) KMT2AEPHX2CASP3FABP5FABP7
SCHEMBL608622 0.84 KMT2A (0.71) KMT2AEPHX2CASP3FABP5FABP7
SCHEMBL17664987 0.84 KMT2A (0.53) KMT2AEPHX2CASP3
SCHEMBL3757636 0.82 KMT2A (0.72) KMT2AEPHX2CASP3FABP5FABP7
SCHEMBL29792075 0.82 KMT2A (0.90) KMT2AEPHX2CASP3FABP5FABP7
SCHEMBL178801 0.82 KMT2A (0.90) KMT2AEPHX2CASP3FABP5FABP7
SCHEMBL29370234 0.82 KMT2A (0.90) KMT2AEPHX2CASP3FABP5FABP7
SCHEMBL7113144 0.81 KMT2A (0.75) KMT2AEPHX2CASP3FABP5FABP7
SCHEMBL1853371 0.81 KMT2A (0.64) KMT2AEPHX2CASP3FABP5FABP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649613-B1 Integrin inhibitors MERCK PATENT GMBH (DE) 2003-11-18 US disclosed
EP-1194401-B1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2003-09-10 EP disclosed
EP-1194401-A1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001005753-A1 DIACYLHYDRAZINE DERIVATIVES MERCK PATENT GMBH (DE) 2001-01-25 WO disclosed