Diftrifmeouron

Diftrifmeouron

SCHEMBL7104017

O=C(NC(=O)c1c(F)cccc1F)Nc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 6/20 0.63
TDP1 Q9NUW8 1/20 0.62
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
GAA P10253 1/20 0.52
FAAH O00519 1/20 0.51
MAPT P10636 2/20 0.51
MEN1 O00255 1/20 0.51
TP53 P04637 1/20 0.51
CASP3 P42574 1/20 0.51
HTT P42858 1/20 0.51
KMT2A Q03164 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
SENP7 Q9BQF6 1/20 0.51
TRPV1 Q8NER1 3/20 0.50
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
MAPK1 P28482 1/20 0.49
EPHX1 P07099 2/20 0.49
STING1 Q86WV6 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9325701 0.97 EPHX2 (0.60) EPHX2TDP1NPC1RAB9AGAA
SCHEMBL11345029 0.91 TDP1 (0.69) EPHX2TDP1NPC1RAB9AGAA
SCHEMBL11246531 0.90 TDP1 (0.52) EPHX2TDP1NPC1RAB9AGAA
SCHEMBL7108246 0.90 MEN1 (0.53) EPHX2TDP1NPC1RAB9AGAA
SCHEMBL10795425 0.87 TDP1 (0.51) EPHX2TDP1NPC1RAB9AGAA
SCHEMBL11319143 0.87 MAPT (0.60) EPHX2TDP1MAPTTRPV1ALDH1A1
SCHEMBL11560696 0.87 EPHX2 (0.60) EPHX2TDP1NPC1RAB9AGAA
SCHEMBL9651342 0.87 MEN1 (0.48) EPHX2TDP1NPC1RAB9AGAA
SCHEMBL10707659 0.86 MEN1 (0.50) EPHX2TDP1NPC1RAB9AGAA
SCHEMBL11026869 0.86 MEN1 (0.53) EPHX2TDP1NPC1RAB9AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE32418-E INSECTICIDES THE DOW CHEMICAL COMPANY (US) 1987-05-12 US claimed
EP-0107214-A2 Pharmaceutical compositions containing benzoyl-phenyl ureas with anti-tumour activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1984-05-02 EP claimed
US-4170657-A INSECTICIDES THE DOW CHEMICAL COMPANY (US) 1979-10-09 US claimed
US-4139636-A N-Phenyl-N'-benzoyl-ureas and pesticidal compositions and uses therefor BAYER AKTIENGESELLSCHAFT (DE) 1979-02-13 US claimed
US-4089975-A DIPHENYL ACYLUREA DERIVATIVE THE DOW CHEMICAL COMPANY (US) 1978-05-16 US claimed
CN-102177905-B 1-(4-trifluoromethoxybenzene)-3-(2,6-difluorobenzoyl) urea preparation TONGHUA PESTICIDE CHEMICAL CO LTD 2013-07-17 CN disclosed
CN-102177905-B 1-(4-trifluoromethoxybenzene)-3-(2,6-difluorobenzoyl) urea preparation TONGHUA PESTICIDE CHEMICAL CO LTD 2013-07-17 CN disclosed
CN-102177905-A 1-(4-trifluoromethoxybenzene)-3-(2,6-difluorobenzoyl) urea preparation TONGHUA PESTICIDE CHEMICAL CO LTD 2011-09-14 CN disclosed
CN-102177904-A Compound preparation of 1-[4-(trifluoromethoxy)phenyl]-3-(2,6-difluorobenzoyl)urea and chlorantraniliprole TONGHUA PESTICIDE CHEMICAL CO LTD 2011-09-14 CN disclosed
CN-102177905-A 1-(4-trifluoromethoxybenzene)-3-(2,6-difluorobenzoyl) urea preparation TONGHUA PESTICIDE CHEMICAL CO LTD 2011-09-14 CN disclosed
CN-102177904-A Compound preparation of 1-[4-(trifluoromethoxy)phenyl]-3-(2,6-difluorobenzoyl)urea and chlorantraniliprole TONGHUA PESTICIDE CHEMICAL CO LTD 2011-09-14 CN disclosed
EP-0917822-B1 Method to control animal ecto-parasites SUMITOMO CHEMICAL CO (JP) 2003-10-08 EP disclosed
EP-0368285-A2 Improved pesticidal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1990-05-16 EP disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
EP-0193249-A2 Benzoyl urea derivatives having ati-tumor activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1986-09-03 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed
EP-0107214-A2 Pharmaceutical compositions containing benzoyl-phenyl ureas with anti-tumour activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1984-05-02 EP disclosed
US-4438110-A 1-(MONO-SUBSTITUTED PHENYL)-3-BENZOYL UREA AND A PHOSPHOROUS CONTAINING COMPOUND UNION CARBIDE CORPORATION (US) 1984-03-20 US disclosed
US-4431667-A Imino ethers useful for controlling insect and arachnoid pests THE UPJOHN COMPANY (US) 1984-02-14 US disclosed
US-4089975-A DIPHENYL ACYLUREA DERIVATIVE THE DOW CHEMICAL COMPANY (US) 1978-05-16 US disclosed