SCHEMBL7106232

SCHEMBL7106232

COC(=O)c1cn(Cc2ccc(C#N)cc2)cc1Cc1cccc(C#N)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
MRGPRX4 Q96LA9 1/20 0.42
AR P10275 1/20 0.42
KLKB1 P03952 2/20 0.41
KLK1 P06870 2/20 0.41
ADRA1D P25100 1/20 0.40
KDM4E B2RXH2 2/20 0.40
IDH1 O75874 1/20 0.39
LMNA P02545 2/20 0.39
HTT P42858 2/20 0.39
RAB9A P51151 1/20 0.39
BRD4 O60885 1/20 0.39
ERCC1 P07992 1/20 0.39
ERCC4 Q92889 1/20 0.39
GRIA2 P42262 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
SNCA P37840 1/20 0.38
GLS O94925 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6170882 0.90 MAPT (0.45) KLKB1KLK1ADRA1DIDH1LMNA
SCHEMBL7101788 0.89 LMNA (0.41) CYP11B1CYP11B2ARKLKB1KLK1
SCHEMBL6163869 0.85 POLB (0.45) CYP11B1CYP11B2KLKB1KLK1ADRA1D
SCHEMBL6165876 0.85 MAPT (0.39) KLKB1KLK1ADRA1DIDH1LMNA
SCHEMBL7102332 0.85 KLKB1 (0.39) CYP11B1CYP11B2KLKB1KLK1ADRA1D
SCHEMBL6163207 0.84 TSHR (0.46) KDM4EIDH1LMNAGRIA2GRIN1
SCHEMBL6164552 0.84 BRD4 (0.50) CYP11B1CYP11B2KLKB1KLK1ADRA1D
SCHEMBL7105719 0.84 POLB (0.47) CYP11B1CYP11B2KLKB1KLK1ADRA1D
SCHEMBL6166642 0.84 KLKB1 (0.42) KLKB1KLK1IDH1LMNABRD4
SCHEMBL7105122 0.84 KLKB1 (0.39) CYP11B1CYP11B2KLKB1KLK1ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030065176-A1 Factor xa inhibitors with aryl-amidines and derivatives, and prodrugs thereof LG CHEM INVESTMENT LTD. (KR) 2003-04-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030065176-A1 Factor xa inhibitors with aryl-amidines and derivatives, and prodrugs thereof F2, F12, TFPI CYP11B1 556/4885CYP11B2 617/4885MRGPRX4 2267/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.