SCHEMBL7115606

SCHEMBL7115606

N#Cc1ccc(CCN2CCN(c3nc4c(OC(N)=O)cccc4[nH]3)CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.49
KCNH2 Q12809 5/20 0.45
KCNJ1 P48048 4/20 0.45
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
HTR1A P08908 1/20 0.38
DRD4 P21917 1/20 0.38
HTR2A P28223 1/20 0.38
HRH1 P35367 1/20 0.38
OPRM1 P35372 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7106768 0.97 PARP1 (0.47) PARP1KCNH2KCNJ1ADRA1DADRA1A
SCHEMBL6871167 0.89 PARP1 (0.43) PARP1HTR1A
SCHEMBL6872714 0.89 PARP1 (0.47) PARP1HTR1AHTR2A
SCHEMBL6875540 0.88 PARP1 (0.42) PARP1ADRA1DADRA1AADRA1B
SCHEMBL6869611 0.88 PARP1 (0.43) PARP1ADRA1DADRA1AADRA1B
SCHEMBL6864442 0.88 PARP1 (0.42) PARP1HTR1AHTR2A
SCHEMBL6871454 0.88 PARP1 (0.42) PARP1ADRA1DADRA1AADRA1BHTR1A
SCHEMBL5621936 0.87 PARP1 (0.65) PARP1
SCHEMBL6875052 0.86 PARP1 (0.49) PARP1KCNH2KCNJ1ADRA1DADRA1A
SCHEMBL6872890 0.86 PARP1 (0.41) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed