SCHEMBL6875540

SCHEMBL6875540

NC(=O)Oc1cccc2[nH]c(N3CCN(CCc4ccc(Cl)cc4)CC3)nc12

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.42
THRB P10828 1/20 0.40
CYP3A4 P08684 1/20 0.40
ABCC1 P33527 1/20 0.40
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
SIGMAR1 Q99720 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6864807 0.96 PARP1 (0.40) PARP1THRBCYP3A4ABCC1SIGMAR1
SCHEMBL6872714 0.91 PARP1 (0.47) PARP1CYP3A4ABCC1
SCHEMBL6871167 0.91 PARP1 (0.43) PARP1CYP3A4ABCC1
SCHEMBL6871454 0.91 PARP1 (0.42) PARP1THRBCYP3A4ABCC1ADRA1D
SCHEMBL6869611 0.91 PARP1 (0.43) PARP1ADRA1DADRA1AADRA1B
SCHEMBL6864442 0.91 PARP1 (0.42) PARP1CYP3A4ABCC1
SCHEMBL6875052 0.89 PARP1 (0.49) PARP1ADRA1DADRA1AADRA1BSIGMAR1
SCHEMBL7115606 0.88 PARP1 (0.49) PARP1ADRA1DADRA1AADRA1B
SCHEMBL6872890 0.88 PARP1 (0.41) PARP1CYP3A4ABCC1
SCHEMBL6869630 0.88 PARP1 (0.41) PARP1CYP3A4ABCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1133477-B1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS ABBOTT GMBH & CO KG (DE) 2004-02-18 EP disclosed