SCHEMBL7116242

SCHEMBL7116242

CC(C)Nc1nc2c(F)c(F)c(Cl)cc2n1[C@@H]1O[C@H](C)[C@@H](O)[C@H]1O

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.55
HSPA8 P11142 1/20 0.39
TRPV4 Q9HBA0 15/20 0.35
ADORA3 P0DMS8 1/20 0.34
FBP1 P09467 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7114592 0.93 HDAC6 (0.54) HDAC6HSPA8TRPV4ADORA3
SCHEMBL7115138 0.89 HDAC6 (0.47) HDAC6HSPA8ADORA3FBP1
SCHEMBL7739904 0.85 HDAC6 (0.63) HDAC6HSPA8TRPV4ADORA3
SCHEMBL7740697 0.85 HDAC6 (0.54) HDAC6HSPA8TRPV4ADORA3FBP1
SCHEMBL7215020 0.84 HDAC6 (0.74) HDAC6HSPA8TRPV4ADORA3FBP1
SCHEMBL7215024 0.84 HDAC6 (0.74) HDAC6HSPA8TRPV4ADORA3FBP1
SCHEMBL10308324 0.84 HDAC6 (0.74) HDAC6HSPA8TRPV4ADORA3FBP1
SCHEMBL7117899 0.81 HDAC6 (0.41) HDAC6TRPV4
SCHEMBL7734307 0.81 HDAC6 (0.49) HDAC6HSPA8TRPV4ADORA3FBP1
SCHEMBL7115561 0.81 HDAC6 (0.60) HDAC6HSPA8TRPV4ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970100-B1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LTD (GB) 2003-11-12 EP claimed
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US claimed
EP-0970100-B1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LTD (GB) 2003-11-12 EP disclosed
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US disclosed