SCHEMBL7119690

SCHEMBL7119690

CC(C)Nc1nc2cc(Cl)c(C(F)(F)F)cc2n1[C@@H]1O[C@H](C)[C@@H](O)[C@H]1O

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.60
HSPA8 P11142 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
ADORA3 P0DMS8 1/20 0.32
CCNT1 O60563 1/20 0.31
CDK9 P50750 1/20 0.31
PTGES O14684 1/20 0.31
SLC15A1 P46059 1/20 0.31
GLP1R P43220 2/20 0.30
DOT1L Q8TEK3 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7115561 0.96 HDAC6 (0.60) HDAC6HSPA8TRPV4ADORA3CCNT1
SCHEMBL7215020 0.88 HDAC6 (0.74) HDAC6HSPA8TRPV4ADORA3CCNT1
SCHEMBL7215024 0.88 HDAC6 (0.74) HDAC6HSPA8TRPV4ADORA3CCNT1
SCHEMBL10308324 0.88 HDAC6 (0.74) HDAC6HSPA8TRPV4ADORA3CCNT1
SCHEMBL7739904 0.85 HDAC6 (0.63) HDAC6HSPA8TRPV4ADORA3CCNT1
SCHEMBL7113212 0.84 HDAC6 (0.62) HDAC6HSPA8ADORA3CCNT1CDK9
SCHEMBL7121805 0.82 HDAC6 (0.45) HDAC6TRPV4PTGES
SCHEMBL7738034 0.82 HDAC6 (0.56) HDAC6HSPA8
SCHEMBL7114052 0.82 HDAC6 (0.49) HDAC6HSPA8TRPV4
SCHEMBL7114288 0.82 HDAC6 (0.49) HDAC6HSPA8TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970100-B1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LTD (GB) 2003-11-12 EP claimed
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US claimed
EP-0970100-B1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LTD (GB) 2003-11-12 EP disclosed
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US disclosed
EP-0970100-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 2000-01-12 EP disclosed
WO-1998035977-A1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 1998-08-20 WO disclosed