SCHEMBL7114288

SCHEMBL7114288

CC(C)Nc1nc2ccc(C(F)(F)F)cc2n1[C@@H]1O[C@H](C)[C@@H](O)[C@H]1O

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.49
MCHR1 Q99705 1/20 0.40
TRPV4 Q9HBA0 2/20 0.37
S1PR1 P21453 3/20 0.36
EGFR P00533 1/20 0.35
CYP11B2 P19099 2/20 0.35
MAT2A P31153 1/20 0.35
HSPA8 P11142 1/20 0.34
IDH1 O75874 2/20 0.34
CYP11B1 P15538 1/20 0.34
HTR3A P46098 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7114052 0.92 HDAC6 (0.49) HDAC6MCHR1TRPV4EGFRHSPA8
SCHEMBL7742258 0.84 HDAC6 (0.57) HDAC6HSPA8HTR3A
SCHEMBL7739725 0.84 CYP11B2 (0.38) EGFRCYP11B2HSPA8CYP11B1HTR3A
SCHEMBL7119690 0.82 HDAC6 (0.60) HDAC6TRPV4HSPA8
SCHEMBL7115561 0.82 HDAC6 (0.60) HDAC6TRPV4HSPA8IDH1
SCHEMBL7738034 0.81 HDAC6 (0.56) HDAC6CYP11B2HSPA8CYP11B1
SCHEMBL7733484 0.81 HDAC6 (0.49) HDAC6TRPV4CYP11B2HSPA8IDH1
SCHEMBL7117206 0.80 HDAC6 (0.48) HDAC6MCHR1TRPV4IDH1
SCHEMBL7215020 0.79 HDAC6 (0.74) HDAC6TRPV4HSPA8
SCHEMBL10308324 0.79 HDAC6 (0.74) HDAC6TRPV4HSPA8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970100-B1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LTD (GB) 2003-11-12 EP claimed
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US claimed
EP-0970100-B1 BENZIMIDAZOLE DERIVATIVES GLAXO GROUP LTD (GB) 2003-11-12 EP disclosed
US-6413938-B1 HERPES VIRUS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2002-07-02 US disclosed