SCHEMBL7120299

SCHEMBL7120299

O=C([C@H](Cc1ccc(OS(=O)(=O)c2cccc3cnccc23)cc1)NS(=O)(=O)c1cccc2cnccc12)N1CCNCC1

nearest known ligand 0.78

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 19/20 0.78
ALDH1A1 P00352 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
LMNA P02545 1/20 0.56
MAPT P10636 1/20 0.56
HTT P42858 1/20 0.56
CAMK2D Q13557 1/20 0.56
P2RX4 Q99571 1/20 0.56
CAMK2A Q9UQM7 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9483456 1.00 P2RX7 (0.78) P2RX7ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL9484593 0.88 P2RX7 (0.87) P2RX7ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL9484591 0.88 P2RX7 (0.87) P2RX7ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL29565839 0.88 P2RX7 (1.00) P2RX7ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL9483837 0.88 P2RX7 (1.00) P2RX7ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL9483834 0.88 P2RX7 (1.00) P2RX7ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL9483968 0.85 P2RX7 (0.72) P2RX7ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL9483973 0.85 P2RX7 (0.72) P2RX7ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL9483789 0.84 P2RX7 (0.76) P2RX7ALDH1A1SMN1; SMN2LMNAMAPT
SCHEMBL9483786 0.84 P2RX7 (0.76) P2RX7ALDH1A1SMN1; SMN2LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003047515-A2 P2X7 RECEPTOR ANTAGONISTS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2003-06-12 WO disclosed
US-5245034-A Compound having vessel smooth muscle relaxation activity Hidaka, Kiroyoshi (JP) 1993-09-14 US disclosed
US-5216150-A Muscle relaxant; enzyme inhibitor and platelet aggutination inhibitor Hidaka, Hiroyoshi (JP) 1993-06-01 US disclosed