SCHEMBL7121335

SCHEMBL7121335

CCc1ccc2c(c1)CC(=O)N2.CCc1ccc2c(c1)CC(=O)N2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.56
PARP1 P09874 1/20 0.51
MAOB P27338 3/20 0.51
GRIA1 P42261 2/20 0.50
CACNG8 Q8WXS5 2/20 0.50
PDE3B Q13370 1/20 0.50
PDE3A Q14432 1/20 0.50
KIF11 P52732 1/20 0.49
PDK2 Q15119 1/20 0.48
SMYD3 Q9H7B4 2/20 0.48
EPHX2 P34913 2/20 0.47
PGR P06401 1/20 0.46
HTR1A P08908 1/20 0.44
DRD2 P14416 1/20 0.44
ADRA1D P25100 1/20 0.44
HTR2A P28223 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP11B1 P15538 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL578518 1.00 AHR (0.56) AHRPARP1MAOBGRIA1CACNG8
SCHEMBL7349900 0.86 AHR (0.53) AHRMAOBGRIA1CACNG8PDE3B
SCHEMBL4509576 0.86 AHR (0.56) AHRPARP1MAOBGRIA1CACNG8
SCHEMBL8670836 0.85 AHR (0.59) AHRMAOBGRIA1CACNG8PDE3B
SCHEMBL2056365 0.84 KIF11 (0.66) PARP1MAOBPDE3BPDE3AKIF11
SCHEMBL12670856 0.84 PARP1 (0.57) AHRPARP1MAOBGRIA1CACNG8
SCHEMBL689189 0.83 AHR (0.50) AHRMAOBGRIA1CACNG8PDE3B
SCHEMBL1460158 0.82 AHR (0.49) AHRMAOBGRIA1CACNG8PDE3B
SCHEMBL12125841 0.82 PARP1 (0.46) AHRPARP1MAOBGRIA1CACNG8
SCHEMBL24570672 0.82 AHR (0.61) AHRMAOBGRIA1CACNG8PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1007505-B1 CERTAIN 5-ALKYL-2-ARYLAMINOPHENYLACETIC ACIDS AND DERIVATIVES NOVARTIS AG (CH) 2003-04-16 EP disclosed