SCHEMBL7121997

SCHEMBL7121997

COc1cc(C(C#N)(CCC(=O)O)C(C)C)cc(OC)c1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 10/20 0.52
CYP3A4 P08684 7/20 0.51
TSHR P16473 3/20 0.51
LMNA P02545 3/20 0.51
KCNH2 Q12809 3/20 0.51
MAPK1 P28482 3/20 0.51
HTR1A P08908 3/20 0.51
HTR2C P28335 3/20 0.51
CACNA1F O60840 2/20 0.51
ADRA2A P08913 2/20 0.51
DRD2 P14416 2/20 0.51
ADRA2C P18825 2/20 0.51
HTR2A P28223 2/20 0.51
SLC6A4 P31645 2/20 0.51
DRD3 P35462 2/20 0.51
SCN1A P35498 2/20 0.51
HTR2B P41595 2/20 0.51
CACNA1D Q01668 2/20 0.51
PDE4D Q08499 2/20 0.51
CACNA1S Q13698 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7132572 0.86 CYP3A4 (0.63) ABCB1CYP3A4TSHRLMNAKCNH2
SCHEMBL7751300 0.86 CYP3A4 (0.63) ABCB1CYP3A4TSHRLMNAKCNH2
SCHEMBL10709109 0.81 ABCB1 (0.55) ABCB1CYP3A4TSHRLMNAKCNH2
SCHEMBL19539141 0.80 ABCB1 (0.60) ABCB1CYP3A4TSHRLMNAKCNH2
SCHEMBL7267395 0.79 ABCB1 (0.59) ABCB1CYP3A4TSHRLMNAKCNH2
SCHEMBL9037850 0.79 ABCB1 (0.59) ABCB1CYP3A4TSHRLMNAKCNH2
SCHEMBL7266275 0.79 ABCB1 (0.59) ABCB1CYP3A4TSHRLMNAKCNH2
SCHEMBL7123218 0.79 NPC1 (0.45) ABCB1CYP3A4TSHRLMNAKCNH2
SCHEMBL11659004 0.79 ABCB1 (0.51) ABCB1CYP3A4TSHRLMNAKCNH2
SCHEMBL10711175 0.77 ABCB1 (0.52) ABCB1CYP3A4TSHRLMNAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6667412-B1 Carboxylic acid, ester or alcohol derivatives; n,n-substi-tuted cyclic amine or phenylacetonitrile intermediates; low cost; stability, workability, final product purity EISAI CO., LTD. (JP) 2003-12-23 US claimed
EP-1167348-A1 NITRILE DERIVATIVES Eisai Co., Ltd. (JP) 2002-01-02 EP claimed
US-6667412-B1 Carboxylic acid, ester or alcohol derivatives; n,n-substi-tuted cyclic amine or phenylacetonitrile intermediates; low cost; stability, workability, final product purity EISAI CO., LTD. (JP) 2003-12-23 US disclosed
EP-1167348-A1 NITRILE DERIVATIVES Eisai Co., Ltd. (JP) 2002-01-02 EP disclosed